Overview

Dabigatran in an Interaction Probe Drug Cocktail

Status:
Completed
Trial end date:
2017-06-01
Target enrollment:
Participant gender:
Summary
Four periods of oral dosing following overnight fasting (1. known metabolic probe drug cocktail consisting of caffeine, diclofenac, esomeprazole, metoprolol, midazolam; 2. dabigatran + cocktail; 3. dabigatran alone; 4. clarithromycin 3 days + cocktail + dabigatran). Blood samples collected for pharmacokinetics over 24 h. Washout between periods. Adverse events, haematology and clinical chemistry recorded.
Phase:
Phase 1
Details
Lead Sponsor:
Turku University Hospital
Treatments:
Caffeine
Clarithromycin
Dabigatran
Diclofenac
Esomeprazole
Metoprolol
Midazolam