Overview

Combination of Olaparib and Navitoclax in Women With HGSC and TNBC

Status:
Not yet recruiting
Trial end date:
2025-04-28
Target enrollment:
Participant gender:
Summary
The purpose of this Phase I study is to determine if the PARP inhibitor olaparib can be safely combined with navitoclax, an inhibitor of Bcl-2/Bcl-XL, in women with TNBC who have somatic or germline mutations in breast cancer gene one (BRCA1) and breast cancer gene two (BRCA2) BRCA1/2 or PALB2 and in women with recurrent HGSC who have progressed greater than 6 months since their last platinum containing chemotherapy. The trial is designed as an open- label multi-center Phase I interventional and translational study. It will identify the dose-limiting toxicities (DLTs), maximum tolerated dose (MTD) and RP2D of olaparib combined with navitoclax for study in Phase II. There is a plan for a follow on Phase II study depending on the results obtained during this Phase I trial.The rationale for this study is that for a subset of patients, olaparib, will increase tumor cell survival dependence on inhibition of cell death by Bcl 2/Bcl- XL. Thus, navitoclax will augment apoptosis induced by PARP inhibition with olaparib.
Phase:
Phase 1
Details
Lead Sponsor:
Sunnybrook Health Sciences Centre
Collaborators:
Centre hospitalier de l'Université de Montréal (CHUM)
Exactis Innovation
Princess Margaret Hospital, Canada
Treatments:
Navitoclax
Olaparib